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Beta-1 adrenergic receptor
URI:
https://gptkb.org/entity/Beta-1_adrenergic_receptor
GPTKB entity
Statements (51)
Predicate
Object
gptkbp:instanceOf
gptkb:protein
gptkb:G_protein-coupled_receptor
gptkbp:alternativeName
gptkb:β1-adrenergic_receptor
gptkb:β1AR
gptkb:beta-1_adrenoceptor
gptkbp:discoveredBy
gptkb:Robert_Lefkowitz
gptkbp:EC_number
7.6.2.1
gptkbp:encodedBy
gptkb:ADRB1_gene
gptkbp:enemyOf
gptkb:atenolol
gptkb:metoprolol
gptkb:acebutolol
gptkb:betaxolol
gptkb:bisoprolol
gptkb:carvedilol
gptkb:dobutamine
gptkb:isoproterenol
gptkb:labetalol
gptkb:nebivolol
propranolol
esmolol
gptkbp:Entrez_Gene_ID
153
gptkbp:expressedIn
gptkb:cardiac_myocytes
gptkb:juxtaglomerular_cells
gptkbp:foundIn
gptkb:human
mammals
gptkbp:function
increases heart rate
increases cardiac contractility
mediates effects of adrenaline and noradrenaline
stimulates renin release
gptkbp:HGNC_ID
gptkb:ADRβ1
https://www.w3.org/2000/01/rdf-schema#label
Beta-1 adrenergic receptor
gptkbp:locatedIn
gptkb:kidney
heart
adipose tissue
gptkbp:locatedOnChromosome
10q25.3
gptkbp:modulatedBy
gptkb:catecholamines
phosphorylation
desensitization
gptkbp:OMIM
109630
gptkbp:receptorSubtype
gptkb:beta-adrenergic_receptor
gptkbp:recipient
adrenergic receptor
gptkbp:significance
involved in heart failure
involved in hypertension
target for beta blockers
gptkbp:structure
seven transmembrane domains
gptkbp:type
activates adenylate cyclase
activates protein kinase A
increases cAMP
gptkbp:UniProtID
P08588
gptkbp:bfsParent
gptkb:CHEMBL1401
gptkbp:bfsLayer
6