|
gptkbp:instanceOf
|
gptkb:adrenergic_receptor
gptkb:G_protein-coupled_receptor
|
|
gptkbp:activatedBy
|
norepinephrine
epinephrine
|
|
gptkbp:associatedWith
|
gptkb:arrhythmia
heart failure
hypertension
|
|
gptkbp:discoveredBy
|
gptkb:Robert_Lefkowitz
|
|
gptkbp:encodedBy
|
gptkb:ADRB1_gene
|
|
gptkbp:enemyOf
|
gptkb:beta_blocker
gptkb:atenolol
gptkb:metoprolol
gptkb:dobutamine
gptkb:isoproterenol
|
|
gptkbp:foundIn
|
gptkb:adipose_tissue
gptkb:kidney
heart
|
|
gptkbp:function
|
increases heart rate
increases cardiac contractility
stimulates renin release
|
|
gptkbp:locatedOn
|
gptkb:plasma_membrane
|
|
gptkbp:locatedOnChromosome
|
chromosome 10q25.3
|
|
gptkbp:orthologIn
|
β2-adrenergic receptor
β3-adrenergic receptor
|
|
gptkbp:structure
|
7 transmembrane domains
|
|
gptkbp:targetOfDrug
|
antiarrhythmic drugs
antihypertensive drugs
|
|
gptkbp:type
|
activates adenylate cyclase
increases cAMP
|
|
gptkbp:UniProtID
|
P08588
|
|
gptkbp:bfsParent
|
gptkb:Beta-1_adrenergic_receptor
|
|
gptkbp:bfsLayer
|
8
|
|
https://www.w3.org/2000/01/rdf-schema#label
|
β1-adrenergic receptor
|