REV-ERB agonist SR9001

GPTKB entity

Statements (23)
Predicate Object
gptkbp:instanceOf REV-ERB agonist
synthetic compound
gptkbp:administeredBy mice
gptkbp:CASNumber 1379686-29-9
gptkbp:chemicalClass benzoxazepine derivative
gptkbp:compatibleWith human use
gptkbp:developedBy gptkb:Scripps_Research_Institute
gptkbp:effect reduced fat mass
improved exercise capacity
increased energy expenditure
https://www.w3.org/2000/01/rdf-schema#label REV-ERB agonist SR9001
gptkbp:mechanismOfAction REV-ERB nuclear receptor agonism
gptkbp:modulatedBy metabolism
circadian rhythm
gptkbp:relatedTo SR9009
gptkbp:routeOfAdministration oral
gptkbp:studiedBy obesity
inflammation
metabolic disorders
gptkbp:target gptkb:REV-ERBα
gptkb:REV-ERBβ
gptkbp:bfsParent gptkb:SR_90001
gptkbp:bfsLayer 8