Tasimelteon

GPTKB entity

Statements (27)
Predicate Object
gptkbp:instanceOf gptkb:drug
melatonin receptor agonist
gptkbp:approvalYear 2014
gptkbp:approvedBy gptkb:FDA
gptkbp:ATCCode N05CH03
gptkbp:brand Hetlioz
gptkbp:CASNumber 609799-22-6
gptkbp:developer gptkb:Vanda_Pharmaceuticals
gptkbp:eliminationHalfLife 1.3 hours
gptkbp:excretion urine
feces
gptkbp:hasMolecularFormula C15H19NO2
https://www.w3.org/2000/01/rdf-schema#label Tasimelteon
gptkbp:legalStatus prescription only
gptkbp:mechanismOfAction MT1 and MT2 melatonin receptor agonist
gptkbp:metabolism liver (CYP1A2, CYP3A4, CYP2C19)
gptkbp:pregnancyCategory C
gptkbp:routeOfAdministration oral
gptkbp:sideEffect headache
elevated liver enzymes
upper respiratory tract infection
nightmares
gptkbp:synonym BMS-214778
gptkbp:usedFor sleep disorders
non-24-hour sleep-wake disorder
gptkbp:bfsParent gptkb:MT1_receptor
gptkbp:bfsLayer 7