AM251

GPTKB entity

Statements (23)
Predicate Object
gptkbp:instanceOf gptkb:chemical_compound
gptkbp:CASNumber 6832-69-7
gptkbp:chemicalFormula C22H25ClN4O
gptkbp:drugClass inverse agonist at CB1 receptor
gptkbp:effect modulates neurotransmitter release
affects memory and learning in animal models
suppresses appetite in animal studies
gptkbp:heldBy cannabinoid receptor antagonist
https://www.w3.org/2000/01/rdf-schema#label AM251
gptkbp:IUPACName 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
gptkbp:legalStatus not approved for medical use
gptkbp:molecularWeight 380.91 g/mol
gptkbp:PubChem_CID CHEMBL127
3083545
gptkbp:relatedTo gptkb:SR141716A
gptkb:rimonabant
gptkbp:routeOfAdministration experimental
gptkbp:studiedBy gptkb:pharmacy
neuroscience
gptkbp:target gptkb:CB1_receptor
gptkbp:UNII 6LR8C1B0AG
gptkbp:bfsParent gptkb:CB1_receptor
gptkbp:bfsLayer 7