nelotanserin

GPTKB entity

Statements (23)
Predicate Object
gptkbp:instanceOf gptkb:chemical_compound
gptkb:drug
gptkbp:CASNumber 337916-20-0
gptkbp:clinicalTrialPhase Phase II
gptkbp:developedBy gptkb:Axovant_Sciences
gptkb:Eli_Lilly_and_Company
gptkbp:hasMolecularFormula C23H29FN2O2
gptkbp:hasSMILES CN1CCC(CC1)N(C)CC(C2=CC=C(F)C=C2)C3=CC4=C(C=C3)OCCO4
https://www.w3.org/2000/01/rdf-schema#label nelotanserin
gptkbp:intendedUse treatment of insomnia
treatment of Parkinson's disease psychosis
gptkbp:IUPACName (2R)-1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-2-(4-fluorophenyl)-N-methyl-N-(1-methylpiperidin-4-yl)ethanamine
gptkbp:mechanismOfAction 5-HT2C receptor antagonist
5-HT2A receptor antagonist
gptkbp:PubChem_CID 11519436
CHEMBL2103882
gptkbp:routeOfAdministration oral
gptkbp:status development discontinued
gptkbp:synonym EMD-281014
RVT-101
gptkbp:UNII 6Q1K1VJ0ZC
gptkbp:bfsParent gptkb:Axovant_Sciences
gptkbp:bfsLayer 7