Relugolix

GPTKB entity

Statements (34)
Predicate Object
gptkbp:instanceOf gptkb:drug
gonadotropin-releasing hormone receptor antagonist
gptkbp:approvalYear 2020
gptkbp:approvedBy gptkb:FDA
gptkb:EMA
gptkbp:ATCCode L02BX07
gptkbp:brand gptkb:Orgovyx
gptkb:Relumina
gptkbp:CASNumber 737789-87-6
gptkbp:chemicalFormula C29H27F2N7O5
gptkbp:developer gptkb:Takeda_Pharmaceutical_Company
gptkb:Myovant_Sciences
gptkbp:eliminationHalfLife 36-65 hours
https://www.w3.org/2000/01/rdf-schema#label Relugolix
gptkbp:KEGGID D10813
gptkbp:legalStatus prescription only
gptkbp:mechanismOfAction suppresses production of testosterone and estrogen
gptkbp:metabolism liver
gptkbp:molecularWeight 602.6 g/mol
gptkbp:pregnancyCategory not recommended
gptkbp:PubChem_CID CHEMBL2103887
46216313
DB15181
gptkbp:routeOfAdministration oral
gptkbp:sideEffect fatigue
increased risk of blood clots
hot flashes
gptkbp:UNII 6Z5B6HVF6O
gptkbp:usedFor prostate cancer
endometriosis
uterine fibroids
gptkbp:bfsParent gptkb:Myovant_Sciences
gptkb:ROIV
gptkbp:bfsLayer 6