|
gptkbp:instanceOf
|
local anesthetic
|
|
gptkbp:ATCCode
|
N01BB03
|
|
gptkbp:boilingPoint
|
389.6 °C
|
|
gptkbp:CASNumber
|
96-88-8
|
|
gptkbp:category
|
amide-type local anesthetic
|
|
gptkbp:chemicalFormula
|
C15H22N2O
|
|
gptkbp:contraindication
|
hypersensitivity to amide anesthetics
|
|
gptkbp:discoveredBy
|
gptkb:Astra_AB
|
|
gptkbp:eliminationHalfLife
|
1.9 to 3.2 hours
|
|
gptkbp:excretion
|
gptkb:kidney
|
|
https://www.w3.org/2000/01/rdf-schema#label
|
Mepivacaine
|
|
gptkbp:introducedIn
|
1957
|
|
gptkbp:IUPACName
|
(RS)-N-(2,6-dimethylphenyl)-1-methyl-piperidine-2-carboxamide
|
|
gptkbp:legalStatus
|
prescription only
|
|
gptkbp:mechanismOfAction
|
blocks sodium channels
|
|
gptkbp:meltingPoint
|
77–78 °C
|
|
gptkbp:metabolism
|
liver
|
|
gptkbp:molecularWeight
|
246.35 g/mol
|
|
gptkbp:pregnancyCategory
|
C
|
|
gptkbp:PubChem_CID
|
CHEMBL1201207
4062
DB00961
|
|
gptkbp:routeOfAdministration
|
injection
|
|
gptkbp:sideEffect
|
allergic reaction
cardiovascular toxicity
central nervous system toxicity
|
|
gptkbp:solubility
|
slightly soluble in water
|
|
gptkbp:synonym
|
Carbocaine
Scandonest
|
|
gptkbp:UNII
|
UQN4C7R3LU
|
|
gptkbp:usedFor
|
local anesthesia
|
|
gptkbp:bfsParent
|
gptkb:Mafeisan_(anesthetic)
|
|
gptkbp:bfsLayer
|
7
|