Aristada

E597293

Aristada is a long-acting injectable antipsychotic medication (aripiprazole lauroxil) used primarily to treat schizophrenia in adults.

All labels observed (2)

Label Occurrences
Aristada canonical 2
Aristada Initio 2

How this entity was disambiguated

Statements (49)

Predicate Object
instanceOf atypical antipsychotic
brand name drug
long-acting injectable antipsychotic medication
approvalYearUS 2015
approvedBy U.S. Food and Drug Administration
ATCCode N05AX12 (aripiprazole)
availableStrength 1064 mg
441 mg
662 mg
882 mg
commonAdverseEffect akathisia
anxiety
injection site pain
insomnia
weight gain
countryApprovedIn United States
dosingInterval every 4 weeks
every 6 weeks
every 8 weeks
formulation extended-release injectable suspension
hasActiveIngredient aripiprazole lauroxil
hasBoxedWarning increased mortality in elderly patients with dementia-related psychosis
hasLoadingDoseOption true
indicatedFor schizophrenia in adults
injectionSite deltoid muscle (for some doses)
gluteal muscle
isLongActing true
isProdrugOf aripiprazole
legalStatusUS prescription only
loadingRegimenBrand Aristada Initio
linked to: Aristada
marketingAuthorizationHolder Alkermes plc
linked to: Alkermes
metabolism CYP2D6
CYP3A4
notApprovedFor treatment of dementia-related psychosis
oralOverlapDrug oral aripiprazole
oralOverlapDuration 21 days (for most initiation regimens)
pharmacologicClass dopamine D2 receptor partial agonist
serotonin 5-HT1A receptor partial agonist
serotonin 5-HT2A receptor antagonist
pregnancyCategoryUS not assigned (use only if benefit justifies risk)
requiresOralOverlap true
routeOfAdministration intramuscular injection
seriousAdverseEffect leukopenia
neuroleptic malignant syndrome
orthostatic hypotension
seizures
tardive dyskinesia
targetPopulation adults with schizophrenia
therapeuticArea psychiatry

How these facts were elicited

Referenced by (4)

Full triples — surface form annotated when it differs from this entity's canonical label.

Alkermes product Aristada
Alkermes product Aristada Initio
linked to: Aristada
Alkermes plc notableProduct Aristada
subject linked to: ALKS
Aristada loadingRegimenBrand Aristada Initio
linked to: Aristada